Velmupressin(Synonyms: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2)

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Velmupressin;(Synonyms: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2)

Velmupressin (c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2) 是一种有效选择性的、短效肽的 V2 受体 (V2R) 激动剂，对 hV2R 和 rV2R 的 EC50 值分别为 0.07 和 0.02 nM。

Velmupressinamp;;(Synonyms: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2)

Velmupressin Chemical Structure

CAS No. : 1647119-61-6

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生物活性

Velmupressin (c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2) is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively[1].

IC50 Target

EC50: 0.07 nM (hV2R), 0.02 nM (rV2R)[1]
分子量

946.58

Formula

C42H60ClN11O8S2
CAS 号

1647119-61-6
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Wiśniewski K, et al. Discovery of Potent, Selective, and Short-Acting Peptidic V2 Receptor Agonists. J Med Chem. 2019 May 23;62(10):4991-5005.