[Sar9,Met(O2)11]-Substance P TFA; 纯度: 99.68%
[Sar9,Met(O2)11]-Substance P TFA 是一种选择性的速激肽 NK1 受体激动剂。
[Sar9,Met(O2)11]-Substance P TFA Chemical Structure
规格 | 价格 | 是否有货 | 数量 |
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1 mg | ¥990 | In-stock | |
5 mg | ¥3900 | In-stock | |
10 mg | ¥6900 | In-stock | |
25 mg | ¥14000 | In-stock | |
50 mg | ; | 询价 | ; |
100 mg | ; | 询价 | ; |
* Please select Quantity before adding items.
[Sar9,Met(O2)11]-Substance P TFA 相关产品
bull;相关化合物库:
- Bioactive Compound Library Plus
- Peptide Library
生物活性 |
[Sar9,Met(O2)11]-Substance P TFA is a tachykinin NK1 receptor selective agonist. |
IC50 Target |
NK1 receptor[1] |
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体外研究 (In Vitro) |
[Sar9,Met(O2)11]-Substance P and septide (10-100 pmol per rat, i.c.v.) are equipotent in increasing mean arterial blood pressure (MAP) and heart rate (HR), yet they have dissimilar time-course. Both agonists increase dose-dependently face washing and sniffing while [Sar9,Met(O2)11]-Substance P is the sole to produce grooming[1]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
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分子量 |
1507.68 |
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Formula |
C66H101N18F3O17S |
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Sequence |
Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-{Sar}-Leu-Met[O2]-NH2 |
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Sequence Shortening |
RPKPQQFF-{Sar}-LM[O2]-NH2 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
Sealed storage, away from moisture
*In solvent : -80deg;C, 6 months; -20deg;C, 1 month (sealed storage, away from moisture) |
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溶解性数据 |
In Vitro:;
H2O : 100 mg/mL (66.33 mM; Need ultrasonic) 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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