c(phg-isoDGR-(NMe)k)

生化分析试剂 Biochemical Assay Reagents
c(phg-isoDGR-(NMe)k);

c(phg-isoDGR-(NMe)k) 是有效选择性的 α5β1 整合素 配体,IC50 为 2.9 nM。

c(phg-isoDGR-(NMe)k)

c(phg-isoDGR-(NMe)k) Chemical Structure

CAS No. : 1844830-65-4

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1 mg ¥5500 询问价格 货期
5 mg ¥9800 询问价格 货期
10 mg ¥15000 询问价格 货期

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c(phg-isoDGR-(NMe)k) 的其他形式现货产品:

c(phg-isoDGR-(NMe)k) TFA

生物活性

c(phg-isoDGR-(NMe)k) is a selective and potent α5β1-integrin ligand with an IC50 of 2.9 nM[1].

IC50 Target

IC50: 2.9 nM (α5β1)[1]

体内研究
(In Vivo)

c(phg-isoDGR-(NMe)k) is trimerized with the chelator TRAP and used as a positron-emission tomography tracer for monitoring α5β1 integrin expression in a M21 mouse xenograft[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

603.67

Formula

C27H41N9O7

CAS 号

1844830-65-4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

参考文献
  • [1]. Kapp TG, et al. N-Methylation of isoDGR Peptides: Discovery of a Selective α5β1-Integrin Ligand as a Potent Tumor Imaging Agent. J Med Chem. 2018 Mar 22;61(6):2490-2499.