天然产物 糖类和糖苷 Saccharides and Glycosides
Rhodionin;(Synonyms: 草质素苷) 纯度: 98.04%
Rhodionin 是从红景天 (Rhodiola crenulata) 的根中分离的,一种特异性非竞争性细胞色素 P450 2D6 抑制剂,IC50 为 0.761 μM,Ki 为 0.769 μM。Rhodionin 有效的,剂量依赖性抑制乙酰胆碱酯酶 (AChE),IC50 范围为 57.50 至 2.43 μg/mL。Rhodionin 具有有效的 DPPH 自由基清除活性,IC50 为 19.49 μM。
Rhodionin Chemical Structure
CAS No. : 85571-15-9
规格 | 价格 | 是否有货 | 数量 |
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10;mM;*;1 mL in DMSO | ¥3314 | In-stock | |
5 mg | ¥3360 | In-stock | |
10 mg | ¥5710 | In-stock | |
50 mg | ; | 询价 | ; |
100 mg | ; | 询价 | ; |
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Rhodionin 相关产品
bull;相关化合物库:
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生物活性 |
Rhodionin, isolated from the root of Rhodiola crenulata, is a specific non-competitive cytochrome P450 2D6 inhibitor with an IC50 of 0.761 μM and a Ki of 0.769 μM[1]. Rhodionin exhibits potent, dose-dependent inhibitory effects on acetylcholinesterase (AChE) with IC50 ranged from 57.50 to 2.43 μg/mL[2]. Rhodionin exhibits potent DPPH free radical scavenging activities, with an IC50 of 19.49 μM[3]. |
IC50 Target |
IC50: 0.761 μM (cytochrome P450 2D6)[1];57.50-2.43 μg/mL (AChE)[2];19.49 μM (DPPH free radical scavenging)[3] |
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分子量 |
448.38 |
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Formula |
C21H20O11 |
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CAS 号 |
85571-15-9 |
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中文名称 |
草质素苷 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
4deg;C, protect from light *In solvent : -80deg;C, 6 months; -20deg;C, 1 month (protect from light) |
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溶解性数据 |
In Vitro:;
DMSO : 16.67 mg/mL (37.18 mM; Need ultrasonic) 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 In Vivo:
请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照 In Vitro 方式配制澄清的储备液,再依次添加助溶剂: ——为保证实验结果的可靠性,澄清的储备液可以根据储存条件,适当保存;体内实验的工作液,建议您现用现配,当天使用; 以下溶剂前显示的百
*以上所有助溶剂都可在 MCE 网站选购。
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参考文献 |
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