Scyliorhinin II;
Scyliorhinin II 是一种选择性的神经激肽-3 (neurokinin-3 tachykinin) 受体激动剂，对大鼠脑皮层的 neurokinin-3 受体的 Ki 值为 2.5 nM。
Scyliorhinin II Chemical Structure
CAS No. : 112748-19-3
| 规格 | 价格 | 是否有货 | |
|---|---|---|---|
| 1 mg | ￥1200 | 询问价格 货期 | |
| 5 mg | ￥2600 | 询问价格 货期 | |
| 10 mg | ￥4200 | 询问价格 货期 | |
| 25 mg | ￥8400 | 询问价格 货期 | |
* Please select Quantity before adding items.
| 生物活性 |
Scyliorhinin II is a selective neurokinin-3 receptor agonist, with a Ki of 2.5 nM for neurokinin-3 receptor in rat cerebral cortex. |
IC50 Target |
Ki: 2.5 nM (Neurokinin-3 receptor)[1] |
|---|---|
| 体外研究 (In Vitro) |
Scyliorhinin II is a neurokinin-3 selective tachykinin receptor, with a Ki of 2.5 nM for neurokinin-3 (NK-3) receptor in rat cerebral cortex. Scyliorhinin II has little effect on NK-1 and NK-2 receptors, with Ki (NK-1 receptor)/Ki (NK-3 receptor) and Ki (NK-2 receptor)/Ki (NK-3 receptor) of 176 and 200[1]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
| 体内研究 (In Vivo) |
Scyliorhinin II produces potent, dose-related reciprocal hindlimb scratching about equipotently with an ED50 of 0.08 nmol via intracerebroventricularly (i.c.v.) administration in mice[2]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
| 分子量 |
1851.09 |
| Formula |
C77H119N21O26S3 |
| CAS 号 |
112748-19-3 |
| Sequence |
Ser-Pro-Ser-Asn-Ser-Lys-Cys-Pro-Asp-Gly-Pro-Asp-Cys-Phe-Val-Gly-Leu-Met-NH2 |
| Sequence Shortening |
SPSNSKCPDGPDCFVGLM-NH2 |
| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
| 参考文献 |
|