Dynorphin A TFA(Synonyms: 肌啡肽A)

Dynorphin A TFA;(Synonyms: 肌啡肽A)

Dynorphin A TFA 是一种内源性阿片肽,是一种高效的 kappa 阿片受体 (KOR) 激活剂。Dynorphin A TFA 也作为其他阿片受体的激动剂,如 mu (MOR) 和 delta (DOR)。

Dynorphin A TFAamp;;(Synonyms: 肌啡肽A)

Dynorphin A TFA Chemical Structure

规格 是否有货
100 mg ; 询价 ;
250 mg ; 询价 ;
500 mg ; 询价 ;

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Dynorphin A TFA 的其他形式现货产品:

Dynorphin A

生物活性

Dynorphin A TFA, an endogenous opioid peptide, is a highy potent kappa opioid receptor (KOR) activator. Dynorphin A TFA also serve as an agonist for other opioid receptors,  such as mu (MOR) and delta (DOR)[1].

IC50 Target

Human Endogenous Metabolite

;

分子量

2261.50

Formula

C101H156F3N31O25

Sequence

Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Trp-Asp-Asn-Gln

Sequence Shortening

YGGFLRRIRPKLKWDNQ

中文名称

肌啡肽A

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

参考文献
  • [1]. Zhang, et al.Dynorphin A as a Potential Endogenous Ligand for Four Members of the Opioid Receptor Gene Family. J Pharmacol Exp Ther. 1998 Jul;286(1):136-41.