PKG inhibitor peptide TFA

发表于由

PKG inhibitor peptide TFA;

PKG inhibitor peptide TFA 是一种 ATP 竞争性的 PKG 抑制剂，Ki 值为 86 μM。

PKG inhibitor peptide TFAamp;;

PKG inhibitor peptide TFA Chemical Structure

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PKG inhibitor peptide TFA 的其他形式现货产品:

PKG inhibitor peptide

生物活性

PKG inhibitor peptide TFA is an ATP-competitive inhibitor of cGMP-dependent protein kinase (PKG), with a Ki of 86 μM[1].

IC50 Target

Ki: 86 μM (PKG)[1]
体外研究
(In Vitro)

Summary of experiments showing that intracellular dialysis of postsynaptic cells with PKG inhibitor PKG inhibitor peptide TFA (1 mM) failed to alter the induction of long-term depression (CCh-LTD)[2].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

1057.13

Formula

C40H75F3N18O12
Sequence

Arg-Lys-Arg-Ala-Arg-Lys-Glu
Sequence Shortening

RKRARKE
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Bhatnagar D, et al. Synthetic peptide analogues differentially alter the binding affinities of cyclic nucleotide dependent protein kinases for nucleotide substrates. Biochemistry. 1988 Mar 22;27(6):1988-94.