hMC1R agonist 1;
hMC1R agonist 1 是一种有效的选择性 hMC1R 激动剂(EC50=3 nM),hMC1R agonist 1 对 hMC1R 的选择性是 hMC3R (b>EC50=902 nM), hMC4R (b>EC50=915 nM), 和 hMC5R (b>EC50=>1000 nM) 的 300 倍。hMC1R agonist 1 有治疗和预防黑皮质素家族疾病的潜能。
hMC1R agonist 1 Chemical Structure
规格 |
|
是否有货 |
|
100 mg |
; |
询价 |
; |
250 mg |
; |
询价 |
; |
500 mg |
; |
询价 |
; |
* Please select Quantity before adding items.
生物活性 |
(EC50=3 nM). hMC1R agonist 1 shows at least 300-fold selectivity for hMC1R over hMC3R (b>EC50=902 nM), hMC4R (b>EC50=915 nM), and hMC5R (b>EC50=>1000 nM). hMC1R agonist 1 has the potential for the therapeutic intervention of melanocortin family[1].
|
IC50 Target |
EC50: 3 nM (hMC1R); 902 nM (hMC3R); 915 nM (hMC4R)[1]
|
分子量 |
|
Formula |
|
运输条件 |
Room temperature in continental US; may vary elsewhere.
|
储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis.
|
参考文献 |
|