Argipressin;(Synonyms: 精氨加压素; Arg8-vasopressin; AVP) 纯度: 99.82%
Argipressin (Arg8-vasopressin) 可与血管精氨酸加压素受体 V1、V2 和 V3 结合,其在 A7r5 大鼠主动脉平滑肌细胞中对 V1 的 Kd 值为 1.31 nM。

Argipressin Chemical Structure
CAS No. : 113-79-1
规格 | 价格 | 是否有货 | 数量 |
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10;mM;*;1 mL in Water | ¥1181 | In-stock | |
1 mg | ¥500 | In-stock | |
5 mg | ¥800 | In-stock | |
10 mg | ¥990 | In-stock | |
25 mg | ¥1200 | In-stock | |
50 mg | ¥1600 | In-stock | |
100 mg | ; | 询价 | ; |
200 mg | ; | 询价 | ; |
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Argipressin 相关产品
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生物活性 |
Argipressin (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1. |
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体外研究 (In Vitro) |
Argipressin binds to the vascular arginine vasopressin receptor, V1, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells. It also stimulates the intracellular release of calcium in A7r5 cells (EC50=5 nM)[1]. AVP-induced [Ca2+]i signals and immunized activity against S-100 in DRG cell culture. The minimum effective concentrations of Argipressin causing [Ca2+]i responses are 100 pM in non-neuronal cells in DRG culture[2]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
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Clinical Trial |
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分子量 |
1084.23 |
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Formula |
C46H65N15O12S2 |
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CAS 号 |
113-79-1 |
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Sequence |
Cys-Tyr-Phe-Gln-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge: Cys1-Cys6) |
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Sequence Shortening |
CYFQNCPRG-NH2 (Disulfide bridge: Cys1-Cys6) |
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中文名称 |
精氨加压素 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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溶解性数据 |
In Vitro:;
H2O : ≥ 100 mg/mL (92.23 mM) * “≥” means soluble, but saturation unknown. 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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