Gluten Exorphin C; 纯度: 98.97%
Gluten exorphin C 是一种源自谷朊粉的阿片肽。在 GPI 和 MVD 检测中,抑制 μ opioid 和 δ opioid 活性,IC50 值分别为 40 μM 和13.5 μM。
Gluten Exorphin C Chemical Structure
CAS No. : 142479-62-7
规格 | 价格 | 是否有货 | 数量 |
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1 mg | ¥1100 | In-stock | |
5 mg | ¥1900 | In-stock | |
10 mg | ¥2900 | In-stock | |
25 mg | ¥5900 | In-stock | |
50 mg | ; | 询价 | ; |
100 mg | ; | 询价 | ; |
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Gluten Exorphin C 相关产品
bull;相关化合物库:
- Bioactive Compound Library Plus
- GPCR/G Protein Compound Library
- Neuronal Signaling Compound Library
- Neurotransmitter Receptor Compound Library
- Anti-Obesity Compound Library
- Peptide Library
生物活性 |
Gluten exorphin C is an opioid peptide derived from wheat gluten. Its IC50 values are 40 μM and 13.5 μM for μ opioid and δ opioid activities in the GPI and MVD assays, respectively. |
IC50 Target |
IC50: 40 μM (μ opioid), 13.5 μM (δ opioid)[1] |
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体外研究 (In Vitro) |
Gluten exorphin C, a novel opioid peptide, is isolated from the pepsin-trypsin-chymotrypsin digest of wheat gluten. Gluten exorphin C is evaluated its opioid activities by the GPI and MVD assays and its receptor affinities by radioreceptor assays. Its IC50s are 40 μM and 13.5 μM in the GPI and the MVD assays, respectively. Gluten exorphin C has a structure quite different from any of the endogenous and exogenous opioid peptides ever reported in that the N terminal Tyr is the only aromatic amino acid. The analogs containing Tyr-Pro-X-Ser-Leu are synthesized to study its structure-activity relationship. Peptides in which X is an aromatic amino acid or an aliphatic hydrophobic amino acid has opioid activity[1]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
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分子量 |
591.70 |
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Formula |
C29H45N5O8 |
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CAS 号 |
142479-62-7 |
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Sequence |
Tyr-Pro-Ile-Ser-Leu |
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Sequence Shortening |
YPISL |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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溶解性数据 |
In Vitro:;
H2O : 100 mg/mL (169.00 mM; Need ultrasonic) 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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