Cyclo(RGDyK)

发表于2023年10月23日由Whatman官网

Cyclo(RGDyK);

Cyclo(RGDyK) 是一种有效的选择性 α_Vβ₃ 整联蛋白 (integrin) 抑制剂，IC₅₀ 为 20 nM。

Cyclo(RGDyK)amp;;

Cyclo(RGDyK) Chemical Structure

CAS No. : 217099-14-4

规格		是否有货
100 mg	;	询价	;
250 mg	;	询价	;
500 mg	;	询价	;

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Cyclo(RGDyK) 的其他形式现货产品:

Cyclo(RGDyK) trifluoroacetate

生物活性	Cyclo(RGDyK) is a potent and selective α_Vβ₃ integrin inhibitor with an IC₅₀ of 20 nM.
IC₅₀ Target	IC50: 20 nM (α_Vβ₃ Integrin), 3000 nM (α_IIbβ₃ Integrin), 4000 nM (α_Vβ₅ Integrin)^[1]
体外研究 (In Vitro)	Cyclo(RGDyK) (c(RGDyK(SAA)) shows high affinity and selectivity for α_Vβ₃ over α_Vβ₅ (IC₅₀=4000 nM) and α_IIbβ₃ (IC₅₀=3000 nM)^[1]. MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量	619.67
Formula	C₂₇H₄₁N₉O₈
CAS 号	217099-14-4
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献	[1]. Haubner R, et al. Glycosylated RGD-containing peptides: tracer for tumor targeting and angiogenesis imaging with improved biokinetics. J Nucl Med. 2001 Feb;42(2):326-36.