Endomorphin 2 TFA(Synonyms: 内吗啡肽 2 三氟乙酸盐)

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Endomorphin 2 TFA (Synonyms: 内吗啡肽 2 三氟乙酸盐) 纯度: 99.55%

Endomorphin 2 TFA，一种高度选择性的高亲和力 μ-opioid 受体激动剂，对 kappa3 结合位点具有高亲和力 ，Ki 为 20 到 30 nM 之间。

Endomorphin 2 TFA (Synonyms: 内吗啡肽 2 三氟乙酸盐)

Endomorphin 2 TFA Chemical Structure

CAS No. : 1276124-00-5

规格 价格 是否有货 数量
10 mM * 1 mL in Water ￥1207 In-stock
5 mg ￥800 In-stock
10 mg ￥1300 In-stock
25 mg ￥2800 In-stock
50 mg   询价  
100 mg   询价  

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Endomorphin 2 TFA 相关产品

•相关化合物库:

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生物活性

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].

IC50 & Target

Ki: 20-30 nM (kappa3 opioid receptor)[1]
分子量

685.69

Formula

C34H38F3N5O7
CAS 号

1276124-00-5
中文名称

内吗啡肽 2 三氟乙酸盐
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Sealed storage, away from moisture

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
溶解性数据
In Vitro: 

H2O : 62.5 mg/mL (91.15 mM; Need ultrasonic)

DMSO : 6 mg/mL (8.75 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 1.4584 mL 7.2919 mL 14.5838 mL
5 mM 0.2917 mL 1.4584 mL 2.9168 mL
10 mM 0.1458 mL 0.7292 mL 1.4584 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.

  • [1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.