Neurokinin A(4-10) TFA; 纯度: 98.10%
Neurokinin A (4-10) TFA 是速激肽 NK2 受体激动剂。
Neurokinin A(4-10) TFA Chemical Structure
| 规格 | 价格 | 是否有货 | 数量 |
|---|---|---|---|
| 1 mg | ￥700 | In-stock | |
| 5 mg | ￥2800 | In-stock | |
| 10 mg | ￥4900 | In-stock | |
| 25 mg | ￥9900 | In-stock | |
| 50 mg | ; | 询价 | ; |
| 100 mg | ; | 询价 | ; |
* Please select Quantity before adding items.
Neurokinin A(4-10) TFA 相关产品
bull;相关化合物库:
- Bioactive Compound Library Plus
- Peptide Library
| 生物活性 |
Neurokinin A (4-10) TFA is a tachykinin NK2 receptor agonist[1]. |
IC50 Target |
NK2 receptor[1] |
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| 体外研究 (In Vitro) |
Neurokinin A (NKA) and its truncated form NKA(4-10) are potent spasmogens of human colon circular muscle, an action mediated exclusively via tachykinin NK2 receptors. A structure-activity study of the neurokinin A (NKA) fragment NKA(4-10) is performed to investigate the importance of amino acid residues for receptor efficacy, potency and affinity at the NK2 receptor in human colon circular muscle. A high density of NK2 receptors has been demonstrated in this tissue, using in vitro autoradiography and radioligand binding[1]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
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| 分子量 |
880.93 |
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| Formula |
C36H55F3N8O12S |
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| Sequence |
Asp-Ser-Phe-Val-Gly-Leu-Met-NH2 |
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| Sequence Shortening |
DSFVGLM-NH2 |
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
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| 储存方式 |
Sealed storage, away from moisture
*In solvent : -80deg;C, 6 months; -20deg;C, 1 month (sealed storage, away from moisture) |
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| 溶解性数据 |
In Vitro:;
H2O : 0.67 mg/mL (0.76 mM; Need ultrasonic) |
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| 参考文献 |
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