Nonapeptide-1 acetate salt(Synonyms: Melanostatine-5 acetate salt)

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Nonapeptide-1 acetate salt;(Synonyms: Melanostatine-5 acetate salt) 纯度: 99.76%

Nonapeptide-1 acetate salt 是一种多肽激素，是强效的 α-黑色素细胞刺激激素 (α-MSH) 的拮抗剂，其 IC50 值为 11 nM。减少黑色素的合成，在很大程度上帮助减少皮肤色素沉着。

Nonapeptide-1 acetate saltamp;;(Synonyms: Melanostatine-5 acetate salt)

Nonapeptide-1 acetate salt Chemical Structure

规格 价格 是否有货 数量
10;mM;*;1 mL in Water ￥4460 In-stock
1 mg ￥800 In-stock
5 mg ￥2200 In-stock
10 mg ￥3200 In-stock
50 mg ; 询价 ;
100 mg ; 询价 ;

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Nonapeptide-1 acetate salt 相关产品

bull;相关化合物库:

  • Bioactive Compound Library Plus
  • GPCR/G Protein Compound Library
  • Neuronal Signaling Compound Library
  • Macrocyclic Compound Library
  • Endocrinology Compound Library
  • Peptide Library

生物活性

Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Reduces synthesis of melanin and helps decrease skin pigmentation to a substantial degree[1].

IC50 Target

IC50: 11 nM (α-MSH)[1].
分子量

1266.56

Formula

C63H91N15O11S
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Sealed storage, away from moisture

Powder -80deg;C 2 years
-20deg;C 1 year

*In solvent : -80deg;C, 6 months; -20deg;C, 1 month (sealed storage, away from moisture)
溶解性数据
In Vitro:;

H2O : 50 mg/mL (39.48 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 0.7895 mL 3.9477 mL 7.8954 mL
5 mM 0.1579 mL 0.7895 mL 1.5791 mL
10 mM 0.0790 mL 0.3948 mL 0.7895 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. Jayawickreme CK, et al. Discovery and structure-function analysis of alpha-melanocyte-stimulating hormone antagonists. J Biol Chem. 1994 Nov 25;269(47):29846-54.