GRK2i TFA

GRK2i TFA; 纯度: 98.13%

GRK2i TFA is a GRK2 inhibitory polypeptide that specifically inhibitsGβγ activation of GRK2. GRK2i TFA corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.

GRK2i TFAamp;;

GRK2i TFA Chemical Structure

规格 价格 是否有货 数量
5 mg ¥5200 In-stock
10 mg ¥8500 In-stock
50 mg ; 询价 ;
100 mg ; 询价 ;

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生物活性

GRK2i TFA is a GRK2 inhibitory polypeptide that specifically inhibitsGβγ activation of GRK2. GRK2i TFA corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.

分子量

3598.10

Formula

C152H257F3N50O43S

Sequence Shortening

WKKELRDAYREAQQLVQRVPKMKNKPRS

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Sealed storage, away from moisture

Powder -80deg;C 2 years
-20deg;C 1 year

*In solvent : -80deg;C, 6 months; -20deg;C, 1 month (sealed storage, away from moisture)

溶解性数据
In Vitro:;

H2O : 100 mg/mL (27.79 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 0.2779 mL 1.3896 mL 2.7792 mL
5 mM 0.0556 mL 0.2779 mL 0.5558 mL
10 mM 0.0278 mL 0.1390 mL 0.2779 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效
储备液的保存方式和期限:-80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)。-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。

参考文献
  • [1]. Jorge A Sierra-Fonseca, et al. Nerve growth factor induces neurite outgrowth of PC12 cells by promoting Gβγ-microtubule interaction. BMC Neurosci. 2014 Dec 31;15:132.