MCH(human, mouse, rat) TFA; 纯度: 99.55%
MCH (human, mouse, rat) TFA 是一种有效的 MCH-R 的肽激动剂，与 MCH1R 和 MCH2R 结合的 IC50 值分别为 0.3 nM 和 1.5 nM。MCH (human, mouse, rat) 对 CHO 细胞系中 MCH-2R 高度敏感，通过 FLIPR 监测细胞内钙动员，显示出功能性激活 MCH-1R 和 MCH-2R 的 EC50 值对分别为 3.9 nM 和 0.1 nM。
MCH(human, mouse, rat) TFA Chemical Structure
| 规格 | 价格 | 是否有货 | 数量 |
|---|---|---|---|
| 5 mg | ￥3500 | In-stock | |
| 10 mg | ￥5900 | In-stock | |
| 50 mg | ; | 询价 | ; |
| 100 mg | ; | 询价 | ; |
* Please select Quantity before adding items.
MCH(human, mouse, rat) TFA 相关产品
bull;相关化合物库:
- Bioactive Compound Library Plus
- Peptide Library
| 生物活性 |
MCH (human, mouse, rat) TFA is a potent peptide agonist of MCH-R and exhibits binding IC50 values of 0.3nM and 1.5 nM for MCH1R and MCH2R, respectively. MCH (human, mouse, rat) is a highly sensitive to MCH-2R in a CHO cell line and monitoring mobilization of intracellular calcium with FLIPR, exhibits functional activation EC50 values of 3.9 nM and 0.1nM for human MCH-1R and MCH-2R, respectively[1]. |
IC50 Target |
Binding IC50: 0.3 nM (MCH1R)IC50: 1.5 nM (MCH1R)[1] |
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| 分子量 |
2500.86 |
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| Formula |
C107H161F3N30O28S4 |
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| Sequence Shortening |
DFDMLRCMLGRVYRPCWQV (Disulfide bridge:Cys7-Cys16) |
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
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| 储存方式 |
Sealed storage, away from moisture
*In solvent : -80deg;C, 6 months; -20deg;C, 1 month (sealed storage, away from moisture) |
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| 溶解性数据 |
In Vitro:;
DMSO : 100 mg/mL (39.99 mM; Need ultrasonic) 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。 In Vivo:
请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照 In Vitro 方式配制澄清的储备液，再依次添加助溶剂： ——为保证实验结果的可靠性，澄清的储备液可以根据储存条件，适当保存；体内实验的工作液，建议您现用现配，当天使用； 以下溶剂前显示的百
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| 参考文献 |
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